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Electrochemical Oxidation of Anastrozole over a BDD Electrode - Role of Operating Parameters and Water Matrix

MetadataDetails
Publication Date2022-11-14
JournalProcesses
AuthorsRebecca Dhawle, Zacharias Frontistis, Dionissios Mantzavinos
InstitutionsUniversity of Patras, University of Western Macedonia
Citations10
AnalysisFull AI Review Included
  • Target Contaminant: The breast-cancer drug Anastrozole (ANZ) was successfully degraded using Electrochemical Oxidation (EO) over a Boron-Doped Diamond (BDD) anode.
  • Performance Benchmark: Maximum ANZ removal reached 97.5% in 90 minutes at the highest tested current density (12.5 mA cm-2).
  • Kinetic Mechanism: Degradation follows pseudo-first-order kinetics, with the rate constant (kapp) doubling from 0.022 to 0.0422 min-1 when the current density was increased from 6.25 to 12.5 mA cm-2.
  • Dominant Oxidant: The primary mechanism relies on electro-generated hydroxyl radicals (¡OH), confirmed by inhibition using tert-butanol. The estimated steady-state concentration of ¡OH was 0.77 x 10-13 M at 12.5 mA cm-2.
  • Matrix Robustness: The EO process is highly robust, maintaining effectiveness across a wide pH range (3-10) and showing only slight reduction in complex matrices (bottled water and wastewater effluent).
  • Chloride Influence: Low chloride concentrations (up to 250 mg L-1) are beneficial due to the generation of secondary oxidants (HOCl, ClO-). However, concentrations above 250 mg L-1 are detrimental due to ¡OH scavenging.
  • Economic Feasibility: The Electric Energy per Order (EEO) ranged from 23.1 to 25 kWh m-3/order, indicating that process economics are highly dependent on electricity costs.
ParameterValueUnitContext
Anode MaterialBoron-Doped Diamond (BDD)B/C = 1000 ppmIdeal non-active electrode
Cathode MaterialStainless SteelN/ACounter electrode
Active Electrode Area16cm2Used for both anode and cathode
Reactor Volume200mLBatch mode operation
Current Density (j) Range6.25 - 12.5mA cm-2Galvanostatic conditions
Initial ANZ Concentration0.5 - 2mg L-1Tested range
Supporting Electrolyte0.1MNa2SO4 (standard) or NaCl
kapp (j = 6.25 mA cm-2)0.0224min-1Inherent pH (6.2)
kapp (j = 12.5 mA cm-2)0.0422min-1Inherent pH (6.2)
kapp (Optimum pH 3)0.0394min-1j = 6.25 mA cm-2
Estimated [¡OH]ss0.77 x 10-13Mj = 12.5 mA cm-2, pH 7
ANZ Diffusion Coefficient3.1 x 10-7cm2/sEstimated via Cottrell equation
EEO Range23.1 - 25kWh m-3/orderCalculated for 6.25 and 12.5 mA cm-2
Cost Estimate3.3 - 3.6€ m-3/orderBased on EU average electricity prices (0.14 €/kWh)
  1. Electrochemical Setup: Experiments were conducted in a 200 mL open plexiglass batch reactor using a BDD anode and a stainless-steel cathode (16 cm2 active area each) under galvanostatic control.
  2. Electrolyte and pH Control: 0.1 M Na2SO4 was used as the standard supporting electrolyte. Initial pH was adjusted (3, 6.2 inherent, 10) using 1 M NaOH or 1 M H2SO4, but the solution was not buffered.
  3. Kinetic Measurement: Samples were collected at timed intervals, immediately quenched with methanol (0.3 mL) to halt radical reactions, filtered, and analyzed using High-Pressure Liquid Chromatography (HPLC) with detection at 210 nm.
  4. Radical Scavenging Test: The role of hydroxyl radicals (¡OH) was confirmed by adding 10 g L-1 of tert-butanol, a known ¡OH scavenger, which resulted in near-complete inhibition of ANZ degradation.
  5. Competition Kinetics: The absolute kinetic constant (kANZ,HO•) and the steady-state concentration of ·OH were estimated using competition kinetics, with Benzoic Acid (BA) serving as the probe compound.
  6. Matrix Evaluation: The process efficiency was tested in three distinct water matrices: ultrapure water (UPW), commercially available bottled water (BW), and secondary treated hospital wastewater effluent (WW).
  7. Economic Analysis: The energy efficiency was quantified using the Electric Energy per Order (EEO) metric, calculated based on power consumption (P), treatment time (t), volume (V), and the apparent rate constant (kapp).
  • Advanced Wastewater Treatment (AWT): BDD EO is highly suitable for tertiary treatment stages in municipal and hospital WWTPs, specifically targeting the removal of persistent organic pollutants (POPs) and emerging contaminants (ECs) like pharmaceuticals (ANZ).
  • Water Reclamation and Reuse: The ability of BDD to achieve high mineralization rates and operate effectively across a wide pH range makes it a robust technology for producing high-quality effluent for industrial or agricultural reuse.
  • Pharmaceutical Manufacturing Effluent: Direct treatment of concentrated pharmaceutical waste streams, where high current densities can be applied to achieve rapid destruction of active pharmaceutical ingredients (APIs).
  • Disinfection and Oxidation: Generation of powerful, non-selective oxidants (¡OH, and active chlorine species in chloride-containing waters) allows for simultaneous disinfection and chemical oxidation of complex organic loads.
  • Industrial Process Water Cleanup: Applicable in industries where water matrices are complex (containing high levels of inorganic ions, bicarbonate, or organic matter) but require reliable contaminant destruction without extensive chemical pre-treatment.
View Original Abstract

The electrochemical oxidation (EO) of the breast-cancer drug anastrozole (ANZ) is studied in this work. The role of various operating parameters, such as current density (6.25 and 12.5 mA cm−2), pH (3-10), ANZ concentration (0.5-2 mg L−1), nature of supporting electrolytes, water composition, and water matrix, have been evaluated. ANZ removal of 82.4% was achieved at 1 mg L−1 initial concentration after 90 min of reaction at 6.25 mA cm−2 and 0.1 M Na2SO4. The degradation follows pseudo-first-order kinetics with the apparent rate constant, kapp, equal to 0.022 min−1. The kapp increases with increasing current density and decreasing solution pH. The addition of chloride in the range 0-250 mg L−1 positively affects the removal of ANZ. However, chloride concentrations above 250 mg L−1 have a detrimental effect. The presence of bicarbonate or organic matter has a slightly negative but not significant effect on the process. The EO of ANZ is compared to its degradation by solar photo-Fenton, and a preliminary economic analysis is also performed.

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